Detalhe da pesquisa
1.
High Prevalence of Plasmodium falciparum K13 Mutations in Rwanda Is Associated With Slow Parasite Clearance After Treatment With Artemether-Lumefantrine.
J Infect Dis
; 225(8): 1411-1414, 2022 04 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-34216470
2.
Efficacy of Cipargamin (KAE609) in a Randomized, Phase II Dose-Escalation Study in Adults in Sub-Saharan Africa With Uncomplicated Plasmodium falciparum Malaria.
Clin Infect Dis
; 74(10): 1831-1839, 2022 05 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-34410358
3.
Insights into the intracellular localization, protein associations and artemisinin resistance properties of Plasmodium falciparum K13.
PLoS Pathog
; 16(4): e1008482, 2020 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-32310999
4.
Artemisinin resistance phenotypes and K13 inheritance in a Plasmodium falciparum cross and Aotus model.
Proc Natl Acad Sci U S A
; 115(49): 12513-12518, 2018 12 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-30455312
5.
Targeting the cell stress response of Plasmodium falciparum to overcome artemisinin resistance.
PLoS Biol
; 13(4): e1002132, 2015 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-25901609
6.
Characterization of Novel Antimalarial Compound ACT-451840: Preclinical Assessment of Activity and Dose-Efficacy Modeling.
PLoS Med
; 13(10): e1002138, 2016 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-27701420
7.
Balancing drug resistance and growth rates via compensatory mutations in the Plasmodium falciparum chloroquine resistance transporter.
Mol Microbiol
; 97(2): 381-95, 2015 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-25898991
8.
Editing the Plasmodium vivax genome, using zinc-finger nucleases.
J Infect Dis
; 211(1): 125-9, 2015 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-25081932
9.
Site-specific genome editing in Plasmodium falciparum using engineered zinc-finger nucleases.
Nat Methods
; 9(10): 993-8, 2012 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-22922501
10.
A conserved metabolic signature associated with response to fast-acting anti-malarial agents.
Microbiol Spectr
; 11(6): e0397622, 2023 Dec 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-37800971
11.
A G358S mutation in the Plasmodium falciparum Na+ pump PfATP4 confers clinically-relevant resistance to cipargamin.
Nat Commun
; 13(1): 5746, 2022 09 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-36180431
12.
Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting Blood-Stage Antimalarial with a High Barrier to Resistance and Potential for Single-Dose Cures in Uncomplicated Malaria.
J Med Chem
; 65(5): 3798-3813, 2022 03 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-35229610
13.
Plasmodium falciparum K13 mutations in Africa and Asia impact artemisinin resistance and parasite fitness.
Elife
; 102021 07 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-34279219
14.
Generation of Transmission-Competent Human Malaria Parasites with Chromosomally-Integrated Fluorescent Reporters.
Sci Rep
; 9(1): 13131, 2019 09 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-31511546
15.
Plasmodium falciparum K13 Mutations Differentially Impact Ozonide Susceptibility and Parasite Fitness In Vitro.
mBio
; 8(2)2017 04 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-28400526
16.
A tetraoxane-based antimalarial drug candidate that overcomes PfK13-C580Y dependent artemisinin resistance.
Nat Commun
; 8: 15159, 2017 05 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-28537265
17.
Artemisinin Action and Resistance in Plasmodium falciparum.
Trends Parasitol
; 32(9): 682-696, 2016 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-27289273
18.
Globally prevalent PfMDR1 mutations modulate Plasmodium falciparum susceptibility to artemisinin-based combination therapies.
Nat Commun
; 7: 11553, 2016 05 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-27189525
19.
Drug resistance. K13-propeller mutations confer artemisinin resistance in Plasmodium falciparum clinical isolates.
Science
; 347(6220): 428-31, 2015 Jan 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-25502314
20.
Genome-wide screen identifies new candidate genes associated with artemisinin susceptibility in Plasmodium falciparum in Kenya.
Sci Rep
; 3: 3318, 2013 Nov 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-24270944